Target of Action

Trenbolone cyclohexylmethylcarbonate, also known as Trenbolone hexahydrobenzylcarbonate, is a synthetic, injected anabolic–androgenic steroid (AAS) of the nandrolone group . It is an androgen ester, specifically the C17β hexahydrobenzylcarbonate (cyclohexylmethylcarbonate) ester of trenbolone . The primary targets of this compound are the androgen receptors in muscle tissues . Buy Trenbolone cyclohexylmethylcarbonate

Mode of Action

This compound acts as a prodrug of trenbolone when administered via intramuscular injection  . It is administered as an ester conjugate to prolong its effective half-life . Once in the bloodstream, plasma lipases cleave the ester group, leaving free trenbolone . This active form of trenbolone then binds to androgen receptors, exerting its anabolic and androgenic effects .

Biochemical Pathways

As an anabolic–androgenic steroid, it likely influences protein synthesis and nitrogen retention in muscle tissues . This leads to increased muscle growth and strength.

Pharmacokinetics

This compound is administered via intramuscular injection . Its ester form allows for a prolonged half-life, ensuring a sustained release of the active compound, trenbolone . The ester group is cleaved by plasma lipases in the bloodstream 

Result of Action

The primary result of this compound’s action is increased muscle growth and appetite . As an anabolic–androgenic steroid, it promotes protein synthesis and nitrogen retention in muscle tissues . This leads to significant increases in muscle mass and strength.

Biochemical Properties

Trenbolone Cyclohexylmethylcarbonate interacts with various enzymes, proteins, and other biomolecules. It is a derivative of nandrolone (19-nortestosterone) and can be bought as parent drug in tablets or as esters such as acetate, enantate, cyclohexylmethylcarbonate, undecylate, or undecanoate in injectable forms .

Cellular Effects

This compound has significant effects on various types of cells and cellular processes. It influences cell function, including any impact on cell signaling pathways, gene expression, and cellular metabolism .

Molecular Mechanism

This compound exerts its effects at the molecular level, including binding interactions with biomolecules, enzyme inhibition or activation, and changes in gene expression .

Temporal Effects in Laboratory Settings

The effects of this compound change over time in laboratory settings. This includes information on the product’s stability, degradation, and any long-term effects on cellular function observed in in vitro or in vivo studies .

Dosage Effects in Animal Models

The effects of this compound vary with different dosages in animal models. This includes any threshold effects observed in these studies, as well as any toxic or adverse effects at high doses .

Metabolic Pathways

This compound is involved in various metabolic pathways, including interactions with enzymes or cofactors. This also includes any effects on metabolic flux or metabolite levels .

Transport and Distribution

This compound is transported and distributed within cells and tissues. This includes any transporters or binding proteins that it interacts with, as well as any effects on its localization or accumulation .

Subcellular Localization

This could include any targeting signals or post-translational modifications that direct it to specific compartments or organelles .

Synthetic Routes and Reaction Conditions

The synthesis of trenbolone hexahydrobenzylcarbonate involves the esterification of trenbolone with hexahydrobenzylcarbonate. The reaction typically requires the use of an acid catalyst and an appropriate solvent. The process involves the following steps:

Preparation of Trenbolone: Trenbolone is synthesized from nandrolone through a series of chemical reactions, including oxidation and reduction steps.

Esterification: Trenbolone is reacted with hexahydrobenzylcarbonate in the presence of an acid catalyst to form trenbolone hexahydrobenzylcarbonate.